Kolb B, Schmid F, Weng J, Altevogt L, Rebelo R.P, Wank B, Baro A, Zens A, Shekhar A, Bilitewski U, Sax S, Wittlin S, Taylor D, Müller R, Laschat S. Total synthesis of tosyl-samroiyotmycin A and its biological profiling. Chemistry. 2024(in press). DOI: 10.1002/chem.202403408

2024
Journal Article
PubMed

Vahekeni N, Brillatz T, Rahmaty M, Cal M, Keller-Märki S, Rocchetti R, Kaiser M, Sax S, Mattli K, Wolfram E, Marcourt L, Queiroz E.F, Wolfender J.L, Mäser P. Antiprotozoal activity of plants used in the management of sleeping sickness in Angola and bioactivity-guided fractionation of Brasenia schreberi J.F.Gmel and Nymphaea lotus L. Active against T. b rhodesiense. Molecules. 2024;29(7):1611. DOI: 10.3390/molecules29071611

2024
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PubMed

Walz A, Sax S, Scheurer C, Tamasi B, Mäser P, Wittlin S. Incomplete Plasmodium falciparum growth inhibition following piperaquine treatment translates into increased parasite viability in the in vitro parasite reduction ratio assay. Front Cell Infect Microbiol. 2024;14:1396786. DOI: 10.3389/fcimb.2024.1396786

2024
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PubMed

Walz A, Duffey M, Aljayyoussi G, Sax S, Leroy D, Besson A, Burrows J.N, Cherkaoui-Rbati M.H, Gobeau N, Westwood M-A, Siethoff C, Gamo S, Mäser P, Wittlin S. The Parasite Reduction Ratio (PRR) assay version 2: standardized assessment of Plasmodium falciparum viability after antimalarial treatment in vitro. Pharmaceuticals (Basel). 2023;16(2):163. DOI: 10.3390/ph16020163

2023
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PubMed

Schalkwijk J, Allman E.L, Jansen P.A.M, de Vries L.E, Verhoef J.M.J, Jackowski S, Botman P.N.M, Beuckens-Schortinghuis C.A, Koolen K.M.J, Bolscher J.M, Vos M.W, Miller K, Reeves S.A, Pett H, Trevitt G, Wittlin S, Scheurer C, Sax S, Fischli C, Angulo-Barturen I, Jimenez-Diaz M.B, Josling G, Kooij T.W.A, Bonnert R, Campo B, Blaauw R.H, Rutjes Fpjt, Sauerwein R.W, Llinas M, Hermkens P.H.H, Dechering K.J. Antimalarial pantothenamide metabolites target acetyl-coenzyme A biosynthesis in Plasmodium falciparum. Sci Transl Med. 2019;11(510):eaas9917. DOI: 10.1126/scitranslmed.aas9917

2019
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PubMed

Massoud M.R, Barry D, Murphy A, Albrecht Y, Sax S, Parchman M. How do we learn about improving health care: a call for a new epistemological paradigm. Int J Qual Health Care. 2016;28(3):420-424. DOI: 10.1093/intqhc/mzw039

2016
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PubMed

Chugh M, Scheurer C, Sax S, Bilsland E, van Schalkwyk D.A, Wicht K.J, Hofmann N, Sharma A, Bashyam S, Singh S, Oliver S.G, Egan T.J, Malhotra P, Sutherland C.J, Beck H.P, Wittlin S, Spangenberg T, Ding X.C. Identification and deconvolution of cross-resistance signals from antimalarial compounds using multidrug-resistant Plasmodium falciparum strains. Antimicrob Agents Chemother. 2015;59(2):1110-1118. DOI: 10.1128/AAC.03265-14

2015
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PubMed

Leven M, Held J, Duffy S, Tschan S, Sax S, Kamber J, Frank W, Kuna K, Geffken D, Siethoff C, Barth S, Avery V.M, Wittlin S, Mordmuller B, Kurz T. Blood schizontocidal and gametocytocidal activity of 3-hydroxy-N'-arylidenepropanehydrazonamides: a new class of antiplasmodial compounds. J Med Chem. 2014;57(19):7971-7976. DOI: 10.1021/jm500811p

2014
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PubMed

Le Manach C, Scheurer C, Sax S, Schleiferböck S, Gonzalez Cabrera D, Younis Y, Paquet T, Street L, Smith P, Ding X, Waterson D, Witty M.J, Leroy D, Chibale K, Wittlin S. Fast in vitro methods to determine the speed of action and the stage-specificity of anti-malarials in Plasmodium falciparum. Malar J. 2013;12:424. DOI: 10.1186/1475-2875-12-424

2013
Journal Article
PubMed